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1Chough Chieyeon, Lee Sunmin, Joung Misuk, Lee Jaemin, Kim Jong Hoon, Kim B. Moon.
Design, synthesis and evaluation of (R)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-5-azaspiro[2.4]heptan-5-yl)-3-oxopropanenitrile as a JAK1-selective inhibitor, MedChemComm, 2018