Results 1 - 10 of 119
- Recent progress toward the asymmetric synthesis of carbon-substituted piperazine pharmacophores and oxidative related heterocycles. Plato A. Magriotis
, RSC Med. Chem.
, 2020
, 11
, 745
- Enantioselective synthesis of gem-disubstituted N-Boc diazaheterocycles via decarboxylative asymmetric allylic alkylation. Alexander W. Sun, Stephan N. Hess, Brian M. Stoltz
, Chem. Sci.
, 2019
, 10
, 788
- Synthesis and evaluation of potent, highly-selective, 3-aryl-piperazinone inhibitors of protein geranylgeranyltransferase-I. Hairuo Peng, Dora Carrico, Van Thai, Michelle Blaskovich, Cynthia Bucher, Erin E. Pusateri, Said M. Sebti, Andrew D. Hamilton
, Org. Biomol. Chem.
, 2006
, 4
, 1768
- Ribose conversion with amino acids into pyrraline platform chemicals – expeditious synthesis of diverse pyrrole-fused alkaloid compounds. Soohyeon Cho, Lina Gu, Ik Joon IN, Bo Wu, Taehoon Lee, Hakwon Kim, Sangho Koo
, RSC Adv.
, 2021
, 11
, 31511
- Synthesis of chiral piperazin-2-ones through palladium-catalyzed asymmetric hydrogenation of pyrazin-2-ols. Guang-Shou Feng, Zi-Biao Zhao, Lei Shi, Yong-Gui Zhou
, Org. Chem. Front.
, 2021
, 8
, 6273
- The hydrophobically-tagged MDM2–p53 interaction inhibitor Nutlin-3a-HT is more potent against tumor cells than Nutlin-3a. Florian Nietzold, Stefan Rubner, Thorsten Berg
, Chem. Commun.
, 2019
, 55
, 14351
- Bifunctional building blocks in the Ugi-azide condensation reaction: a general strategy toward exploration of new molecular diversity. Steven Gunawan, Christopher Hulme
, Org. Biomol. Chem.
, 2013
, 11
, 6036
- Pd-Catalysed asymmetric allylic alkylation of heterocycles: a user's guide. François Richard, Paul Clark, Al Hannam, Thomas Keenan, Alexandre Jean, Stellios Arseniyadis
, Chem. Soc. Rev.
, 2024
, 53
, 1936
- Synthesis of 1- and 4-substituted piperazin-2-ones via Jocic-type reactions with N-substituted diamines. Michael S. Perryman, Matthew W. M. Earl, Sam Greatorex, Guy J. Clarkson, David J. Fox
, Org. Biomol. Chem.
, 2015
, 13
, 2360
- Selective inhibitors of fibroblast activation protein (FAP) with a xanthine scaffold. Koen Jansen, Hans De Winter, Leen Heirbaut, Jonathan D. Cheng, Jurgen Joossens, Anne-Marie Lambeir, Ingrid De Meester, Koen Augustyns, Pieter Van der Veken
, Med. Chem. Commun.
, 2014
, 5
, 1700